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K048
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Synthesis and testing of structural fragments of acetylcholinesterase reactivators - K027 and K048
Publication without faculty affiliation
publication
A comparison of tabun-inhibited rat brain acetylcholinesterase reactivation by three oximes (HI-6, obidoxime, and K048) in vivo detected by biochemical and histochemical techniques
2010 |
Faculty of Medicine in Hradec Králové
publication
Optimalization of the synthesis of new acetylcholinesterase reactivators - K027 and K048
Publication without faculty affiliation
publication
Novel acetylcholinesterase reactivator - oxime K048 - reactivation activity in vitro
2010 |
Central Library of Charles University
publication
A comparison of the efficiacy of new asymmetric bispyridinium oximes (K027, K048) with currently available oximes against tabun by in vivo methods
2006 |
Faculty of Pharmacy in Hradec Králové
publication
In Vivo Evaluation of Cholinesterase Activity, Oxidative Stress Markers, Cyto- and Genotoxicity of K048 Oxime - a Promising Antidote against Organophosphate Poisoning
2014 |
Publication without faculty affiliation
publication
Bisquaternary oximes as reactivators of tabun-inhibited human brain cholinesterases: an in vitro study
2007 |
Publication without faculty affiliation
publication
SAR study in the class of acetylcholinesterase reactivators
Publication without faculty affiliation
publication
Bisquaternary oximes as reactivators of tabun-inhibited human brain cholinesterases: an in vitro study
2007 |
Central Library of Charles University, Faculty of Pharmacy in Hradec Králové
publication
Synthesis of new acetylcholinesterase reactivators. Structural fragments and in vitro evaluation of their biological potency
Publication without faculty affiliation
publication
Comparative determination of the efficacy of bispyridinium oximes in paraoxon poisoning
2015 |
Publication without faculty affiliation
publication
Novel Group of AChE Reactivators-Synthesis, In Vitro Reactivation and Molecular Docking Study
2018 |
Publication without faculty affiliation
publication
In Vitro Evaluation of Oxidative Stress Induced by Oxime Reactivators of Acetylcholinesterase in HepG2 Cells
2023 |
Faculty of Pharmacy in Hradec Králové
publication
Oxidative stress status assessment of rats' brains injury following subacute exposure to K-oximes
2023 |
Publication without faculty affiliation
publication
Butyrylcholinesterase inhibited by nerve agents is efficiently reactivated with chlorinated pyridinium oximes
2019 |
Publication without faculty affiliation
publication
Charged pyridinium oximes with thiocarboxamide moiety are equally or less effective reactivators of organophosphate-inhibited cholinesterases compared to analogous carboxamides
2022 |
Publication without faculty affiliation
publication
Pyridinium oximes with ortho-positioned chlorine moiety exhibit improved physicochemical properties and efficient reactivation of human Acetylcholinesterase inhibited by several nerve agents
2018 |
Publication without faculty affiliation
publication
A review of the synthesis of quaternary Acetylcholinesterase reactivators
2018 |
Publication without faculty affiliation
publication
Pharmacological and toxicological in vitro and in vivo effect of higher doses of oxime reactivators
2019 |
Publication without faculty affiliation