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Search for publications relevant for "peptidomimetics"
peptidomimetics
Publication
Class
Person
Publication
Programmes
publication
On the role of the R configuration of the reaction-intermediate isostere in HIV-1 protease-inhibitor binding: X-ray structure at 2.0 angstrom resolution
2006 |
Faculty of Science
publication
Unorthodox Inhibitors of HIV Protease: Looking Beyond Active-site-directed Peptidomimetics
2014 |
Faculty of Science
publication
Peptidomimetic inhibitors complexed with HIV-1 proteinase: Crystallisation for X-ray diffraction studies.
Publication without faculty affiliation
publication
Aromatic reduced amide bond peptidomimetics as selective inhibitors of neuronal nitric oxide synthase
2003 |
First Faculty of Medicine
publication
Potency comparison of Peptidomimetic Inhibitors against HIV-1 and HIV-2 proteinases: design of equipotent lead compounds
Publication without faculty affiliation
publication
Potency comparison of peptidomimetic inhibitors against HIV-1 and HIV-2 proteinases: design of equipotent lead compounds.
Publication without faculty affiliation
publication
Aromatic reduced amide bond peptidomimetics as selective inhibitors of neuronal nitric oxide synthase
2003 |
Faculty of Physical Education and Sport
publication
Structural determinants for subnanomolar inhibition of the secreted aspartic protease Sapp1p from Candida parapsilosis
2021 |
Faculty of Science
publication
Reduced amide bond peptidomimetics. (4S)-N-(4-amino-5-(aminoalkyl)aminopentyl)-N´-nitroguanidines, potent and highly selective inhibitors of neuronal nitric oxide synthase
2001 |
First Faculty of Medicine
publication
Structure-Activity Relationship of F-18-Labeled Phosphoramidate Peptidomimetic Prostate-Specific Membrane Antigen (PSMA)-Targeted Inhibitor Analogues for PET Imaging of Prostate Cancer
2016 |
Central Library of Charles University
publication
Hydroxyethylamine Isostere of an HIV-1 Protease Inhibitor Prefers Its Amine to the Hydroxy Group in Binding to Catalytic Aspartates. A Synchrotron Study of HIV-1 Protease in Complex with a Peptidomimetic Inhibitor.
2002 |
Faculty of Science
publication
Hydroxyethylamine Isostere of an HIV-1 Protease Inhibitor Prefers Its Amine to the Hydroxy Group in Binding to Catalytic Aspartates. A Synchrotron Study of HIV-1 Protease in Complex with a Peptidomimetic Inhibitor.
2002 |
First Faculty of Medicine, Faculty of Mathematics and Physics
publication
An Activity-Based Probe for Cathepsin K Imaging with Excellent Potency and Selectivity
2021 |
Faculty of Science, Faculty of Physical Education and Sport, Central Library of Charles University
publication
Probing tripodal peptide scaffolds as insulin and IGF-1 receptor ligands
2018 |
Central Library of Charles University
publication
Minimal pharmacophoric elements and fragment hopping, an approach directed at molecular diversity and isozyme selectivity. Design of selective neuronal nitric oxide synthase inhibitors
2008 |
First Faculty of Medicine
publication
Discovery of Highly Potent and Selective Inhibitors of Neuronal Nitric Oxide Synthase by Fragment Hopping
2009 |
First Faculty of Medicine
publication
An ethylenamine inhibitor binds tightly to both wild type and mutant HIV-1 proteases. Structure and energy study.
2003 |
Faculty of Science
publication
An ethylenamine inhibitor binds tightly to both wild type and mutant HIV-1 proteases. Structure and energy study.
2003 |
First Faculty of Medicine, Faculty of Mathematics and Physics
publication
Structural Basis for Inhibition of Cathepsin B Drug Target from the Human Blood Fluke, Schistosoma mansoni
2011 |
Faculty of Science
publication
Structure-activity relationship and biochemical evaluation of novel fibroblast activation protein and prolyl endopeptidase inhibitors with α-ketoamide warheads
2021 |
Faculty of Science, Faculty of Physical Education and Sport, Central Library of Charles University
publication
Structure-activity relationship and biochemical evaluation of novel fibroblast activation protein and prolyl endopeptidase inhibitors with alpha-ketoamide warheads
2021 |
Faculty of Science, Faculty of Physical Education and Sport, Central Library of Charles University
publication
Biomimetic Macrocyclic Inhibitors of Human Cathepsin D: Structure-Activity Relationship and Binding Mode Analysis
2020 |
Faculty of Science, Faculty of Physical Education and Sport
publication
Highly potent inhibitors of cathepsin K with a differently positioned cyanohydrazide warhead: structural analysis of binding mode to mature and zymogen-like enzymes
2022 |
Faculty of Science, Faculty of Physical Education and Sport
publication
Phenotypic screening of the 'Kurz-box' of chemicals identifies two compounds (BLK127 and HBK4) with anthelmintic activity in vitro against parasitic larval stages of Haemonchus contortus
2019 |
Faculty of Pharmacy in Hradec Králové