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acetylcholinesterase inhibition
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A new group of monoquaternary reactivators of acetylcholinesterase inhibited by nerve agents
2005 |
Faculty of Education
publication
In-vitro searching for a new potent reactivator of acetylcholinesterase inhibited by nerve agent VX
2005 |
Publication without faculty affiliation
publication
Reactivation of acetylcholinesterase inhibited by the pesticide chlorpyrifos
2006 |
Faculty of Pharmacy in Hradec Králové, Central Library of Charles University
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Molecular Aspects of the Reactivation Process of Acetylcholinesterase Inhibited by Cyclosarin
2011 |
Publication without faculty affiliation
publication
Acetylcholinesterase-Inhibiting Activity of Salicylanilide N-Alkylcarbamates and Their Molecular Docking
2012 |
Faculty of Pharmacy in Hradec Králové
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Oxime K074-in vitro and in silico reactivation of acetylcholinesterase inhibited by nerve agents and pesticides
2020 |
Publication without faculty affiliation
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Pretreatment with L-Carinitine Enhanced Acetylcholinesterase Inhibition Following Galantamine Administration in Rats
Publication without faculty affiliation
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The effect of L-carnitine pretreatment on acetylcholinesterase inhibition of intracerebroventricularly (i.c.v.) administered 7-methoxytacrine
Publication without faculty affiliation
publication
Reactivation of acetylcholinesterase inhibited with cyclosarine and chlorpyrifos - relationship between structure of reactivators and their reactivation potency
Publication without faculty affiliation
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Molecular modeling and in vitro reactivation study between the oxime BI-6 and acetylcholinesterase inhibited by different nerve agents
2015 |
Publication without faculty affiliation
publication
Molecular Modeling and In Vitro Studies of a Neutral Oxime as a Potential Reactivator for Acetylcholinesterase Inhibited by Paraoxon
2018 |
Faculty of Medicine in Hradec Králové
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Pyridinium oximes with ortho-positioned chlorine moiety exhibit improved physicochemical properties and efficient reactivation of human Acetylcholinesterase inhibited by several nerve agents
2018 |
Publication without faculty affiliation
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In vitro functional interactions of acetylcholine esterase inhibitors and muscarinic receptor antagonists in the urinary bladder of the rat
2014 |
Faculty of Pharmacy in Hradec Králové
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Diethyl 2-(Phenylcarbamoyl)phenyl Phosphorothioates: Synthesis, Antimycobacterial Activity and Cholinesterase Inhibition
2014 |
Faculty of Pharmacy in Hradec Králové
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Multidrug Resistance Modulation Activity of Silybin Derivatives and Their Anti-inflammatory Potential
2020 |
Faculty of Medicine in Pilsen
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Hydrazones of 4-(Trifluoromethyl)benzohydrazide as New Inhibitors of Acetyl- and Butyrylcholinesterase
2021 |
Faculty of Pharmacy in Hradec Králové
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Different inhibition of acetylcholinesterase in selected parts of the rat brain following intoxication with VX and Russian VX
2009 |
First Faculty of Medicine
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N-Alkyl-2-[4-(trifluoromethyl)benzoyl]hydrazine-1-carboxamides and Their Analogues: Synthesis and Multitarget Biological Activity
2020 |
Faculty of Pharmacy in Hradec Králové
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Different sensitivity of miniature endplate currents of the rat extensor digitorum longus, soleus and diaphragm muscles to a novel acetylcholinesterase inhibitor C-547
2006 |
Faculty of Science
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Effect of galantamine on acetylcholinesterase and butyrylcholinesterase activities in the presence of L-carnitine in rat selected brain and peripheral tissues
2006 |
First Faculty of Medicine
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Galantamine antiacetylcholinesterase activity in rat brain influenced by L-carnitine
2005 |
Faculty of Medicine in Hradec Králové
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Analysis of Amarylidaceae alkaloids from Zephyranthes grandiflora by GC/MS and their cholinesterase activity
2011 |
Publication without faculty affiliation
publication
Alkaloids from Zephyranthes robusta Baker and Their Acetylcholinesterase- and Butyrylcholinesterase-Inhibitory Activity
2013 |
Faculty of Pharmacy in Hradec Králové
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Chlorpyrifos-methyl oxon hydrolysis and its monitoring by HPLC-MS/MS
2018 |
Faculty of Science
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UHPLC-HRMS study of pharmacokinetics of a novel hybrid cholinesterase inhibitor K1234: A comparison between in silico, in vitro and in vivo data
2022 |
Faculty of Medicine in Hradec Králové
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Some possibilities to study new prophylactics against nerve agents
2019 |
Publication without faculty affiliation
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Oxime K033-reactivation Activity of Cholinesterases Inhibited by Various Nerve Agents and Organophosphorus Pesticides
2018 |
Publication without faculty affiliation
publication
Effect of cognitive drugs on mitochondrial respiration and activity of electron transport chain complexes
2014 |
First Faculty of Medicine
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Phenothiazine-Tacrine Heterodimers: Pursuing Multitarget Directed Approach in Alzheimer's Disease
2021 |
Publication without faculty affiliation
publication
New hybrids of tacrine and indomethacin as multifunctional acetylcholinesterase inhibitors
2021 |
Faculty of Pharmacy in Hradec Králové