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drug discovery
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publication
The Potential Applications of Artificial Intelligence in Drug Discovery and Development
2021 |
First Faculty of Medicine
publication
Drug Discovery against Cryptosporidium parvum
Publication without faculty affiliation
publication
Future of Drug Discovery: The Synergy of Edge Computing, Internet of Medical Things, and Deep Learning
2023 |
Faculty of Medicine in Pilsen
publication
Drugs discovery in Cryptosporidium parvum
Publication without faculty affiliation
publication
Drug Discovery against Cryptosporidium parvum. Grant Progress Report
Publication without faculty affiliation
publication
The Utilization of the Monte Carlo Technique for Rational Drug Discovery
2016 |
First Faculty of Medicine
publication
Targeted D-4 Dopamine Receptors: Implications for Drug Discovery and Therapeutic Development
2013 |
First Faculty of Medicine, Second Faculty of Medicine
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Drug Discovery against Cryptosporidium parvum. Grant Progress Report 2002
Publication without faculty affiliation
publication
Drug discovery in Cryptosporidium parvum: What we can learn from molecular and biochemical analyses
Publication without faculty affiliation
publication
Blood-brain barrier in vitro models as tools in drug discovery: Assessment of the transport ranking of antihistaminic drugs
2012 |
Faculty of Pharmacy in Hradec Králové
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Sustainable Drug Discovery of Multi-Target-Directed Ligands for Alzheimer's Disease
2021 |
Publication without faculty affiliation
publication
Total Synthesis of Natural Products: Case Studies in the Evaluation of New Synthetic Methods, Structural Elucidation and Drug Discovery
2022 |
Faculty of Science
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ADAMANT: a placebo-controlled randomized phase 2 study of AADvac1, an active immunotherapy against pathological tau in Alzheimer's disease
2021 |
Second Faculty of Medicine
publication
Anti-viral drug discovery against monkeypox and smallpox infection by natural curcumin derivatives: A Computational drug design approach
2023 |
Faculty of Medicine in Hradec Králové
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Re-emerging Aspartic Protease Targets: Examining Cryptococcus neoformans Major Aspartyl Peptidase 1 as a Target for Antifungal Drug Discovery
2021 |
Faculty of Science, Central Library of Charles University
publication
Molpher
Publication without faculty affiliation
publication
Advances in Antifungal Drug Development: An Up-To-Date Mini Review
2021 |
Faculty of Pharmacy in Hradec Králové
publication
Using Bayesian Modeling on Molecular Fragments Features for Virtual Screening
2016 |
Faculty of Mathematics and Physics
publication
Set-up and screening of a fragment library targeting the 14-3-3 protein interface
2019 |
Faculty of Science
publication
Boron cluster compounds as new chemical leads for antimicrobial therapy
2021 |
Faculty of Science
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Novel Aeruginosin-865 from Nostoc sp as a Potent Anti-inflammatory Agent
2013 |
Faculty of Science
publication
Novel sustainable-by-design HDAC inhibitors for the treatment of Alzheimer's disease
2019 |
Publication without faculty affiliation
publication
Synthesis and Cytotoxic and Antiviral Activity Profiling of All-Four Isomeric Series of Pyrido-Fused 7-Deazapurine Ribonucleosides
2020 |
Faculty of Science
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Synthesis of Selagibenzophenone A and Its Derivatives for Evaluation of Their Antiproliferative, ROR gamma Inverse Agonistic, and Antimicrobial Effect
2023 |
Faculty of Science
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Designing and development of phthalimides as potent anti-tubulin hybrid molecules against malaria
2022 |
Faculty of Science
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Small-molecule inhibitors of cyclophilin D as potential therapeutics in mitochondria-related diseases
2022 |
Publication without faculty affiliation
publication
Rational Discovery of GSK3-Beta Modulators Aided by Protein Pocket Prediction and High-Throughput Molecular Docking
2016 |
Publication without faculty affiliation
publication
Turning Donepezil into a Multi-Target-Directed Ligand through a Merging Strategy
2021 |
Publication without faculty affiliation
publication
Pharmaceutical Applications
2017 |
Faculty of Pharmacy in Hradec Králové
publication
High-Throughput Fluorescent Assay for Inhibitor Screening of Proteases from RNA Viruses
2021 |
Central Library of Charles University